<div id="pf1" class="pf w0 h0" data-page-no="1"><div class="pc pc1 w0 h0"><img class="bi x0 y0 w1 h0" alt="" src="https://files.passeidireto.com/5019db8f-e2a0-4f59-8b1e-d68d6768012b/bg1.png"><div class="t m0 x1 h1 y1 ff1 fs0 fc0 sc0 ls1 ws0">CLASSIFICAÇÃO<span class="blank"> </span>DOS<span class="blank"> </span>AGONIST<span class="blank _0"></span>AS<span class="blank"> </span>MUSCARÍNICOS</div><div class="t m0 x2 h2 y2 ff2 fs0 fc0 sc0 ls1 ws1">1.<span class="blank _1"> </span>DROGAS<span class="blank"> </span>DE<span class="blank"> </span>AÇÃO<span class="blank"> </span>DIRET<span class="blank _0"></span>A</div><div class="t m0 x2 h2 y3 ff2 fs0 fc0 sc0 ls1 ws2">\u25cf<span class="blank _2"> </span>ocupam<span class="blank"> </span>e<span class="blank"> </span>ativam<span class="blank"> </span>receptores<span class="blank"> </span>muscarínicos</div><div class="t m0 x3 h2 y4 ff2 fs0 fc0 sc0 ls1 ws3">-<span class="blank _3"> </span>acetilcolina<span class="blank"> </span>(n)</div><div class="t m0 x3 h2 y5 ff2 fs0 fc0 sc0 ls1 ws4">-<span class="blank _3"> </span>betanecol<span class="blank"> </span>(s)</div><div class="t m0 x3 h2 y6 ff2 fs0 fc0 sc0 ls1 ws5">-<span class="blank _3"> </span>carbacol<span class="blank"> </span>(s)</div><div class="t m0 x3 h2 y7 ff2 fs0 fc0 sc0 ls1 ws6">-<span class="blank _3"> </span>pilocarpina<span class="blank"> </span>(n)</div><div class="t m0 x2 h2 y8 ff2 fs0 fc0 sc0 ls1 ws1">2.<span class="blank _1"> </span>DROGAS<span class="blank"> </span>DE<span class="blank"> </span>AÇÃO<span class="blank"> </span>INDIRET<span class="blank _0"></span>A</div><div class="t m0 x2 h2 y9 ff2 fs0 fc0 sc0 ls1 ws7">\u25cf<span class="blank _2"> </span>inibem<span class="blank"> </span>a<span class="blank"> </span>ação<span class="blank"> </span>da<span class="blank"> </span>acetilcolinesterase,<span class="blank"> </span>aumentando<span class="blank"> </span>os<span class="blank"> </span>níveis<span class="blank"> </span>de<span class="blank"> </span>ACh<span class="blank"> </span>e</div><div class="t m0 x4 h2 ya ff2 fs0 fc0 sc0 ls1 ws8">potencializando<span class="blank"> </span>seus<span class="blank"> </span>efeitos.</div><div class="t m0 x1 h1 yb ff1 fs0 fc0 sc0 ls1 ws9">EFEITOS<span class="blank"> </span>DOS<span class="blank"> </span>AG<span class="blank _4"></span>ONIST<span class="blank _0"></span>AS<span class="blank"> </span>MUSCARÍNICOS</div><div class="t m0 x2 h2 yc ff2 fs0 fc0 sc0 ls1 wsa">\u25cf<span class="blank _2"> </span>efeitos<span class="blank"> </span>cardiovasculares:<span class="blank"> </span>diminuição<span class="blank"> </span>da<span class="blank"> </span>frequência<span class="blank"> </span>e<span class="blank"> </span>do<span class="blank"> </span>débito<span class="blank"> </span>cardíaco<span class="blank"> </span>e</div><div class="t m0 x4 h2 yd ff2 fs0 fc0 sc0 ls1 wsb">vasodilatação<span class="blank"> </span>generalizada,<span class="blank"> </span>produzindo<span class="blank"> </span>queda<span class="blank"> </span>da<span class="blank"> </span>pressão<span class="blank"> </span>arterial.</div><div class="t m0 x2 h2 ye ff2 fs0 fc0 sc0 ls1 wsb">\u25cf<span class="blank _2"> </span>efeitos<span class="blank"> </span>sobre<span class="blank"> </span>o<span class="blank"> </span>músculo<span class="blank"> </span>liso:<span class="blank"> </span>contração<span class="blank"> </span>e<span class="blank"> </span>aumento<span class="blank"> </span>do<span class="blank"> </span>peristaltismo<span class="blank"> </span>gastroint.</div><div class="t m0 x4 h2 yf ff2 fs0 fc0 sc0 ls1 wsc">brônquios<span class="blank"> </span>e<span class="blank"> </span>bexiga<span class="blank"> </span>também<span class="blank"> </span>contraem.</div><div class="t m0 x3 h2 y10 ff2 fs0 fc0 sc0 ls1 wsd">-<span class="blank _3"> </span>efeito<span class="blank"> </span>adverso:<span class="blank"> </span>diarreia<span class="blank"> </span>e<span class="blank"> </span>náuseas,<span class="blank"> </span>devido<span class="blank"> </span>ao<span class="blank"> </span>aumento<span class="blank"> </span>do<span class="blank"> </span>peristaltismo.</div><div class="t m0 x3 h2 y11 ff2 fs0 fc0 sc0 ls1 wse">-<span class="blank _3"> </span>efeito<span class="blank"> </span>adverso:<span class="blank"> </span>urgência<span class="blank"> </span>miccional.</div><div class="t m0 x2 h2 y12 ff2 fs0 fc0 sc0 ls1 ws7">\u25cf<span class="blank _2"> </span>efeitos<span class="blank"> </span>sobre<span class="blank"> </span>glândulas:<span class="blank"> </span>sudoríparas,<span class="blank"> </span>lacrimal,<span class="blank"> </span>salivar<span class="blank"> </span>e<span class="blank"> </span>brônquica-<span class="blank"> </span>provocam</div><div class="t m0 x4 h2 y13 ff2 fs0 fc0 sc0 ls1 ws8">estimulação<span class="blank"> </span>de<span class="blank"> </span>glândulas<span class="blank"> </span>exócrinas.</div><div class="t m0 x3 h2 y14 ff2 fs0 fc0 sc0 ls1 ws7">-<span class="blank _3"> </span>efeito<span class="blank"> </span>adverso:<span class="blank"> </span>diaforese,<span class="blank"> </span>suor<span class="blank"> </span>excessivo.</div><div class="t m0 x2 h2 y15 ff2 fs0 fc0 sc0 ls1 wsf">\u25cf<span class="blank _2"> </span>efeitos<span class="blank"> </span>sobre<span class="blank"> </span>o<span class="blank"> </span>olho:<span class="blank"> </span>contração<span class="blank"> </span>do<span class="blank"> </span>músculo<span class="blank"> </span>ciliar<span class="blank _0"></span>.</div><div class="t m0 x3 h2 y16 ff2 fs0 fc0 sc0 ls1 ws7">-<span class="blank _3"> </span>efeito<span class="blank"> </span>adverso:<span class="blank"> </span>miose,<span class="blank"> </span>contração<span class="blank"> </span>das<span class="blank"> </span>pupilas.</div><div class="t m0 x1 h1 y17 ff1 fs0 fc0 sc0 ls1 ws9">USOS<span class="blank"> </span>TERAPÊUTICOS</div><div class="t m0 x2 h1 y18 ff2 fs0 fc0 sc0 ls0">\u25cf<span class="ff1 ls1 ws10">betanecol</span><span class="ls1 ws11">:<span class="blank"> </span>estimula<span class="blank"> </span>o<span class="blank"> </span>músculo<span class="blank"> </span>liso<span class="blank"> </span>do<span class="blank"> </span>TGI<span class="blank"> </span>e<span class="blank"> </span>bexiga<span class="blank"> </span>em<span class="blank"> </span>certos<span class="blank"> </span>quadros<span class="blank"> </span>neurológicos</span></div><div class="t m0 x4 h2 y19 ff2 fs0 fc0 sc0 ls1 ws8">e<span class="blank"> </span>pós-cirúrgicos.<span class="blank"> </span>(m3)</div><div class="t m0 x2 h1 y1a ff2 fs0 fc0 sc0 ls0">\u25cf<span class="ff1 ls1 ws10">pilocarpina</span><span class="ls1 ws7">:<span class="blank"> </span>glaucoma,<span class="blank"> </span>xerostomia<span class="blank"> </span>(boca<span class="blank"> </span>seca)<span class="blank"> </span>(m3)</span></div><div class="t m0 x2 h1 y1b ff2 fs0 fc0 sc0 ls0">\u25cf<span class="ff1 ls1 ws10">cevimelina</span><span class="ls1 ws12">:<span class="blank"> </span>xerostomia.<span class="blank"> </span>(m3)</span></div><div class="t m0 x2 h1 y1c ff2 fs0 fc0 sc0 ls0">\u25cf<span class="ff1 ls1 ws13">agonistas<span class="blank"> </span>m1-seletivos</span><span class="ls1 ws14">:<span class="blank"> </span>em<span class="blank"> </span>estudo<span class="blank"> </span>p/<span class="blank"> </span>alzheimer<span class="blank _0"></span>.</span></div><div class="t m0 x1 h1 y1d ff1 fs0 fc0 sc0 ls1 ws15">CONTRA-<span class="blank"> </span>INDICAÇÕES:</div><div class="t m0 x2 h2 y1e ff2 fs0 fc0 sc0 ls1 ws16">\u25cf<span class="blank"> </span>asmáticos</div><div class="t m0 x2 h2 y1f ff2 fs0 fc0 sc0 ls1 ws17">\u25cf<span class="blank _2"> </span>distúrbios<span class="blank"> </span>pépticos<span class="blank"> </span>ácidos</div><div class="t m0 x2 h2 y20 ff2 fs0 fc0 sc0 ls1 ws16">\u25cf<span class="blank"> </span>hipotensão</div><div class="t m0 x2 h2 y21 ff2 fs0 fc0 sc0 ls1 ws18">\u25cf<span class="blank _2"> </span>insuficiência<span class="blank"> </span>coronariana</div></div><div class="pi" data-data="{"ctm":[1.000000,0.000000,0.000000,1.000000,0.000000,0.000000]}"></div></div> <div id="pf2" class="pf w0 h0" data-page-no="2"><div class="pc pc2 w0 h0"><img class="bi x0 y0 w1 h0" alt="" src="https://files.passeidireto.com/5019db8f-e2a0-4f59-8b1e-d68d6768012b/bg2.png"></div><div class="pi" data-data="{"ctm":[1.000000,0.000000,0.000000,1.000000,0.000000,0.000000]}"></div></div>
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